Epinastine HCl

CAS No. 108929-04-0

Epinastine HCl ( Epinastine Hydrochloride; Alesion; Elestat )

Catalog No. M17804 CAS No. 108929-04-0

Epinastine is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
25MG 45 In Stock
50MG 59 In Stock
100MG 87 In Stock
200MG 165 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Epinastine HCl
  • Note
    Research use only, not for human use.
  • Brief Description
    Epinastine is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.
  • Description
    Epinastine Hydrochloride is a histamine H1 receptor antagonist without sedative activity. Epinastine hydrochloride blocks the histamine H1 receptor and inhibits the release of histamine from mast cells. This prevents the typical allergic symptoms that are caused by histamine activity on capillaries, skin, and mucous membranes. Typical histamine activities include vasodilation, bronchoconstriction, increased vascular permeability, pain, itching, and spasmodic contractions of gastrointestinal smooth muscles. Epinastine HCl also has affinity for histamine H2, 5-HT2, and the alpha-1, alpha-2 adrenergic receptors.
  • Synonyms
    Epinastine Hydrochloride; Alesion; Elestat
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    HT
  • Research Area
    Inflammation/Immunology
  • Indication
    ——

Chemical Information

  • CAS Number
    108929-04-0
  • Formula Weight
    285.77
  • Molecular Formula
    C16H15N3·HCl
  • Purity
    98%
  • Solubility
    ——
  • SMILES
    Cl[H].NC1=NCC2N1C1=CC=CC=C1CC1=CC=CC=C21
  • Chemical Name
    3-Amino-9,13b-dihydro-1H-dibenzo[c,f]imidazo[1,5-a]azepine Hydrochloride

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Fügner A, et al. Arzneimittelforschung, 1988, 38(10), 1446-1453.
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